Found 23 Enz. Inhib. hit(s) with Target = 'Cholecystokinin receptor type A' and Ligand = 'BDBM50005463' 
Affinity DataKi: 0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
Affinity DataKi: 10.4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0794nMAssay Description:Binding affinity against cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Ability to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Concentration required for 50% inhibition of Cholecystokinin type A receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of cholecystokinin A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Half maximal inhibition of specific binding of [125I]-Bolton-Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of binding of [125I]- CCK-33 to rat pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Half-maximal inhibition of [125I]CCK-33 binding to cholecystokinin A receptor from rat pancreatic tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Antagonistic activity against cholecystokinin type A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125 I] CCK-8 from Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of [125I]-Cholecystokinin-8 (125I-CCK-8) binding to Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreas.More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Half-maximal inhibition of specific binding of [125I]bolton hunter CCK-8 to rat pancreas cholecystokinin type A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Binding of [3H]-propionyl-CCK-8 to Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 0.710nMAssay Description:In vitro inhibition of [3H]propionyl-CCK-8 binding to rat pancreatic membranes at Cholecystokinin type A receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 0.710nMAssay Description:Binding affinity by competitive inhibition of the radioligand [3H]pCCK-8 at Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 0.794nMAssay Description:Binding affinity against cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of binding of [125I]-CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A(Cavia porcellus)
Merck Sharp & Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp & Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of binding of [125I]- CCK-33 to guinea pig cortexMore data for this Ligand-Target Pair
