Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Cholecystokinin receptor type A' and Ligand = 'BDBM50343720'
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50343720(3-(4-(5-(4-methoxyphenyl)-4-p-tolylpyrimidine-2-ca...)
Affinity DataIC50:  2nMAssay Description:Displacement of [I125]-CCK8 from human CCK1 receptor expressed in CHO Flip cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50343720(3-(4-(5-(4-methoxyphenyl)-4-p-tolylpyrimidine-2-ca...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human CCK1 receptor expressed in CHO Flip cells assessed as increase of radio labeled inositol phosphate accumulation by Wallac m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed