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Found 1 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 5 activator 1' and Ligand = 'BDBM50340912'
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50340912((4-amino-2-(pyridin-4-ylamino)thiazol-5-yl)(4-fluo...)
Affinity DataIC50:  400nMAssay Description:Inhibition of CDK5/p25 assessed as [33P]gamma-ATP incorporation into peptide PKTPKKAKKL substrate after 45 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed