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Found 2 Enz. Inhib. hit(s) with Target = 'Cysteinyl leukotriene receptor 1' and Ligand = 'BDBM50064079'
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50064079(4-Oxo-2-[3-((E)-2-quinolin-2-yl-vinyl)-phenyl]-4H-...)
Affinity DataIC50:  408nMAssay Description:Antagonist activity at CysLT1 receptor in human dU937 cells assessed as inhibition of LTD4-induced increase of calcium level treated 30 mins before L...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064079(4-Oxo-2-[3-((E)-2-quinolin-2-yl-vinyl)-phenyl]-4H-...)
Affinity DataKd:  408nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed