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Found 4 Enz. Inhib. hit(s) with Target = 'D(1A)/D(2) dopamine receptor' and Ligand = 'BDBM50225361'
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50225361(Etisulergine)
Affinity DataIC50:  25nMAssay Description:Noncompetitive Inhibitory activity against rat striatal synaptosomal DHPR enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50225361(Etisulergine)
Affinity DataIC50:  25nMAssay Description:In vitro inhibitory activity was evaluated against,[3H]spiperone calf caudate (SPC) dopamine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50225361(Etisulergine)
Affinity DataIC50:  120nMAssay Description:In vitro inhibitory activity was evaluated against,[3H]dopamine (DA),calf caudate dopamine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50225361(Etisulergine)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against human liver Dihydrodipicolinate reductase (DHPR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed