Affinity DataKi: 160nMAssay Description:In vitro binding affinity tested on human Dopamine receptor D2 using [3H]spiperon as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:In vitro binding affinity tested on human Dopamine receptor D2 (long) using [3H]spiperon as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+4nMAssay Description:In vitro binding affinity tested on human Dopamine receptor D2 (short) using [3H]spiperone as a radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity at human D2R expressed in HEK293 cells incubated for 3 mins by FLIPR analysisMore data for this Ligand-Target Pair