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Found 3 Enz. Inhib. hit(s) with Target = 'D(3) dopamine receptor' and Ligand = 'BDBM50326734'
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50326734(7-((2-(4-(biphenyl-4-yl)piperazin-1-yl)ethyl)(prop...)
Affinity DataKi:  5.22nMAssay Description:Displacement of [3H]spiperone from rat D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50326734(7-((2-(4-(biphenyl-4-yl)piperazin-1-yl)ethyl)(prop...)
Affinity DataKi:  5.22nMAssay Description:Displacement of [3H]spiperone from rat D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50326734(7-((2-(4-(biphenyl-4-yl)piperazin-1-yl)ethyl)(prop...)
Affinity DataEC50:  1.03nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed