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Found 2 Enz. Inhib. hit(s) with Target = 'DNA gyrase subunit A/B' and Ligand = 'BDBM50197073'
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50197073(3-amino-7-((R)-3-((S)-1-aminoethyl)pyrrolidin-1-yl...)
Affinity DataIC50:  200nMAssay Description:Inhibition of recombinant full-length C-terminal His6-tagged Escherichia coli DNA gyrase AB supercoiling activity using relaxed DNA as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50197073(3-amino-7-((R)-3-((S)-1-aminoethyl)pyrrolidin-1-yl...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Escherichia coli gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed