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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) with Target = 'DNA topoisomerase 1' and Ligand = 'BDBM50142525'
Target
DNA topoisomerase 1
(Homo sapiens (Human))
Kumamoto University
Curated by
ChEMBL
Ligand
BDBM50142525
(CHEMBL47524 | N-(4,5-Dihydro-thiazol-2-yl)-3,4,5-t...)
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Affinity Data
IC50: 3.44E+4nM
Assay Description:
Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed form
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
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