Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membrane measured after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membrane measured after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding affinity was determined towards Opioid receptor delta 1 in rat brain synaptosomes using [3H]-deltorphin II as radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:The compound was tested for the ability to displace opioid receptor kappa specific radioligand [3H]DADLEMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity of Opioid receptor delta 1 by the displacement of delta-selective [3H]DSLET from brain membrane preparations.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:The compound was tested for the ability to displace delta-receptor specific radioligand [3H]DSLETMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Binding affinity against Opioid receptor delta 1 by displacement of radioligand [3H]-DSLET in rat brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Inhibition of [3H]- ]DSLET binding to opioid receptor delta from rat brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]DSLET from Opioid receptor delta 1 from rat brain homogenateMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Binding affinity for Opioid receptor delta 1 determined by displacing [3H]-DSLET from rat brain membrane binding sitesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Binding affinity for delta opioid receptors was determined by displacement of [3H]DSLET from rat brain membrane binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Tested for binding affinity towards Opioid receptor delta 1 in rat and guinea pig brain membrane binding assaysMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Tested for binding affinity against delta opioid receptor by displacing [3H]- DSLET radioligand from rat brain membrane preparationsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataKi: 6nMAssay Description:Binding affinity against Opioid receptor delta 1 of guinea pig brain membranes using 1 nM of [3H]DADLE as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]-deltorphin 2 from delta opioid receptor in rat GH3 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataKi: 6.30nMAssay Description:Inhibition of [3H]-Deltorphin 2 binding to mouse delta opioid receptor expressed in rat GH3 cell membranes by Cheng-Prusoff analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Binding affinity to delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Agonist activity at delta opioid receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataKi: 6.90nMAssay Description:Inhibition of [3H]-Deltorphin 2 binding to mouse delta opioid receptor expressed in HEK293 cell membranes incubated for 60 mins by Cheng-Prusoff anal...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 27.7nMAssay Description:Inhibition of [3H][D-Ala2,D-Leu5]enkephalin binding to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Binding affinity of the compound towards Opioid receptor delta 1 was determined using [d-Ser2, Leu5, Thr6] enkephalin (DSLET) as the radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 1.10nMAssay Description:Agonist activity at FLAG-tagged mouse delta opioid receptor expressed in human HEK293 cells assessed as inhibition of forskolin stimulated cAMP produ...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 1.10nMAssay Description:Agonist activity at FLAG-tagged mouse delta opioid receptor expressed in human HEK293 cells assessed as inhibition of forskolin stimulated cAMP produ...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 1.30nMAssay Description:Agonist activity at mouse FLAG-tagged delta opioid receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP production pre...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 1.40nMAssay Description:Agonist activity at mouse FLAG-tagged delta opioid receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP production pre...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 11nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 11nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 11nMAssay Description:Inhibitory potency against Opioid receptor delta 1 in the mouse vas deferens assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of binding of [3H]naloxone to Opioid receptor mu 1 in the rat brain homogenateMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 22nMAssay Description:In vitro inhibitory activity was determined against Opioid receptor delta 1 in mouse vas deferensMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataEC50: 74nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electric-field induced measured after 5 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO-K1 cells assessed as beta-arrestin2 recruitment incubated for 90 mins by PathHunter ...More data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at human DOR expressed in CHO cells assessed as reduction in ERK1/2 phosphorylation levelMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonist activity at DOP (unknown origin) expressed in SH-SY5Y cell membranes co-expressing Gbeta1-RGFP protein assessed as induction of G protein act...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0800nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0800nMAssay Description:Agonist activity at delta opioid receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells co-expressing beta-arrestin2 assessed as beta-arrestin2 recruitment measured a...More data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Agonist activity at DOP (unknown origin) expressed in SH-SY5Y cell membranes co-expressing beta-arrestin2-RGFP protein assessed as induction of beta-...More data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells co-expressing beta-arrestin2 assessed as beta-arrestin2 recruitment measured a...More data for this Ligand-Target Pair