TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 258nMAssay Description:Displacement of [3H]DSLET from DOR in rat brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+4nMAssay Description:Antagonist activity against delta opioid receptor in mouse vas deference assessed as effect on DPDPE-induced responseMore data for this Ligand-Target Pair