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Found 1 Enz. Inhib. hit(s) with Target = 'Diacylglycerol O-acyltransferase 1' and Ligand = 'BDBM176289'
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM176289(US9688696, 4)
Affinity DataIC50:  407nMpH: 7.4 T: 2°CAssay Description:DGAT activity in membrane preparations was assayed in 50 mM Tris-HCl (pH 7.4), 150 mM MgCl2, 1 mM EDTA and 0.2% BSA, containing 50 μM DAG, 32 &#...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent