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Found 6 Enz. Inhib. hit(s) with Target = 'Dihydroorotate dehydrogenase (quinone), mitochondrial' and Ligand = 'BDBM92602'
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum)
Harvard Medical School

LigandPNGBDBM92602(DHOD Inhibitor, 1 | US8703811, 2)
Affinity DataIC50:  930nMAssay Description:Assay was determined using a continuous assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum)
Harvard Medical School

LigandPNGBDBM92602(DHOD Inhibitor, 1 | US8703811, 2)
Affinity DataIC50:  930nMAssay Description:Type 2 DHODH activity was monitored with either the direct assay measuring the formation of orotate or via a chromogen reduction assay using DCIP. Al...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium vivax)
Genzyme

US Patent
LigandPNGBDBM92602(DHOD Inhibitor, 1 | US8703811, 2)
Affinity DataIC50:  5.60E+3nMAssay Description:Type 2 DHODH activity was monitored with either the direct assay measuring the formation of orotate or via a chromogen reduction assay using DCIP. Al...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium vivax)
Genzyme

US Patent
LigandPNGBDBM92602(DHOD Inhibitor, 1 | US8703811, 2)
Affinity DataIC50:  5.60E+3nMAssay Description:Assay was determined using a continuous assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Genzyme

US Patent
LigandPNGBDBM92602(DHOD Inhibitor, 1 | US8703811, 2)
Affinity DataIC50: >3.00E+4nMAssay Description:Type 2 DHODH activity was monitored with either the direct assay measuring the formation of orotate or via a chromogen reduction assay using DCIP. Al...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Genzyme

US Patent
LigandPNGBDBM92602(DHOD Inhibitor, 1 | US8703811, 2)
Affinity DataIC50: >3.00E+4nMAssay Description:Assay was determined using a continuous assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed