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Found 1 Enz. Inhib. hit(s) with Target = 'Dual specificity tyrosine-phosphorylation-regulated kinase 1A' and Ligand = 'BDBM162328'
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Arrien Pharmaceuticals

US Patent
LigandPNGBDBM162328(US9669028, 77 (6-(3-methyl-1H-pyrazolo[3,4-b]pyrid...)
Affinity DataIC50: >1.00E+3nMpH: 7.5Assay Description:The 2×DYRK1A/Ser/Thr 18 mixture was prepared in 50 mM HEPES pH 7.5, 0.01% BRIJ-35, 10 mM MgCl2, 1 mM EGTA. The final 10 μL Kinase Reaction consi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent