Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'E3 ubiquitin-protein ligase Mdm2' and Ligand = 'BDBM50165717'
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50165717(CHEMBL3799390)
Affinity DataIC50:  1.07E+3nMAssay Description:Binding affinity to human MDM2 assessed as inhibition of interaction with p53 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed