Found 1 Enz. Inhib. hit(s) with Target = 'E3 ubiquitin-protein ligase parkin' and Ligand = 'BDBM562069'
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education and Research
US Patent
Mayo Foundation For Medical Education and Research
US Patent
Affinity DataEC50: 405nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair