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Found 3 Enz. Inhib. hit(s) with Target = 'Endothelin-1 receptor' and Ligand = 'BDBM50029353'
TargetEndothelin-1 receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50029353(CHEMBL414165 | [(5S,8S,11R,14R,16aR)-8-(1H-Indol-3...)
Affinity DataIC50:  1.20nMAssay Description:Inhibitory effect of the compound against Human ET-A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50029353(CHEMBL414165 | [(5S,8S,11R,14R,16aR)-8-(1H-Indol-3...)
Affinity DataIC50:  3nMAssay Description:The compound was tested for binding inhibitory activity against Endothelin A receptor from porcine aortic smooth muscle membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50029353(CHEMBL414165 | [(5S,8S,11R,14R,16aR)-8-(1H-Indol-3...)
Affinity DataIC50:  3nMAssay Description:Inhibitory effect of the compound against porcine ET-A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed