Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'Epidermal growth factor receptor [T790M,L858R]' and Ligand = 'BDBM195873'
TargetEpidermal growth factor receptor [T790M,L858R](Homo sapiens (Human))
East China University of Science and Technology

US Patent
LigandPNGBDBM195873(US9670213, Compound 018 N-(3-(2-(4-morpholinopheny...)
Affinity DataIC50:  3.02nMT: 2°CAssay Description:In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent