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Found 4 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM50364076'
TargetEstrogen receptor(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50364076(CHEMBL198159)
Affinity DataEC50:  286nMAssay Description:Agonist activity at human ERalpha expressed in HEC-1 cells coexpressing beta-gal assessed as luciferase activity after 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50364076(CHEMBL198159)
Affinity DataEC50:  205nMAssay Description:Agonist activity at human ERalpha expressed in U2OS cells coexpressing pCMX-hSRC3 assessed as luciferase activity after 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50364076(CHEMBL198159)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at human N-His6-tagged terbium-labelled NRID-SRC3 of ERalpha ligand binding domain expressed in Escherichia coli BL21 cells after 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50364076(CHEMBL198159)
Affinity DataEC50:  637nMAssay Description:Agonist activity at human N-His6-tagged terbium-labelled ERalpha ligand binding domain expressed in Escherichia coli BL21 cells assessed as recruitme...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed