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Found 2 Enz. Inhib. hit(s) with Target = 'Estrogen receptor beta' and Ligand = 'BDBM50178328'
TargetEstrogen receptor beta(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50178328((3S,10S,13S,17S)-13,17-dimethyl-10-vinyl-2,3,4,7,8...)
Affinity DataIC50:  25nMAssay Description:Binding affinity to human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50178328((3S,10S,13S,17S)-13,17-dimethyl-10-vinyl-2,3,4,7,8...)
Affinity DataEC50:  31nMAssay Description:Effect on transactivation of ALP gene expression in HEK293 cells transfected with hERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed