Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Geranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50076132'
LigandPNGBDBM50076132((S)-4-Methyl-2-({4-[(pyridin-4-ylmethyl)-amino]-bi...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibition of [3H]-GGPP incorporation into H-Ras-CVLL by Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed