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Found 2 Enz. Inhib. hit(s) with Target = 'Ghrelin O-acyltransferase' and Ligand = 'BDBM396236'
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM396236(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of human GOAT expressed in HEK293 cells harboring -preproghrelin in presence of Octanoate-BSA incubated for 5 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM396236(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)
Affinity DataIC50:  0.0200nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent