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Found 2 Enz. Inhib. hit(s) with Target = 'Glucagon receptor' and Ligand = 'BDBM50244337'
TargetGlucagon receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50244337(CHEMBL511964 | trans-4-(((4-tert-butylcyclohexyl)(...)
Affinity DataIC50:  9nMAssay Description:Displacement of [125I]glucagon from human GCGR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50244337(CHEMBL511964 | trans-4-(((4-tert-butylcyclohexyl)(...)
Affinity DataIC50:  23nMAssay Description:Antagonist activity against human GCGR expressed in CHO cells assessed as glucagon-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed