Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with Target = 'Glutamate receptor 3' and Ligand = 'BDBM50060635'
TargetGlutamate receptor 3(RAT)
Sibia Neurosciences

Curated by PDSP Ki Database
LigandPNGBDBM50060635((S)-2-Amino-3-(5-fluoro-2,4-dioxo-3,4-dihydro-2H-p...)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
TargetGlutamate receptor 3(RAT)
Sibia Neurosciences

Curated by PDSP Ki Database
LigandPNGBDBM50060635((S)-2-Amino-3-(5-fluoro-2,4-dioxo-3,4-dihydro-2H-p...)
Affinity DataKi:  70nMAssay Description:Displacement of (R,S)-[5-methyl-3H]AMPA from rat recombinant flop iGluR3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 3(Homo sapiens (Human))
Sibia Neurosciences

Curated by PDSP Ki Database
LigandPNGBDBM50060635((S)-2-Amino-3-(5-fluoro-2,4-dioxo-3,4-dihydro-2H-p...)
Affinity DataKi:  179nMMore data for this Ligand-Target Pair
TargetGlutamate receptor 3(Homo sapiens (Human))
Sibia Neurosciences

Curated by PDSP Ki Database
LigandPNGBDBM50060635((S)-2-Amino-3-(5-fluoro-2,4-dioxo-3,4-dihydro-2H-p...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
TargetGlutamate receptor 3(Homo sapiens (Human))
Sibia Neurosciences

Curated by PDSP Ki Database
LigandPNGBDBM50060635((S)-2-Amino-3-(5-fluoro-2,4-dioxo-3,4-dihydro-2H-p...)
Affinity DataEC50:  2.09E+4nMAssay Description:Agonist activity at recombinant GluA3 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetGlutamate receptor 3(RAT)
Sibia Neurosciences

Curated by PDSP Ki Database
LigandPNGBDBM50060635((S)-2-Amino-3-(5-fluoro-2,4-dioxo-3,4-dihydro-2H-p...)
Affinity DataEC50:  2.09E+4nMAssay Description:Agonist activity at cyclothiazide-desensitized rat recombinant flip iGluR3 expressed in Xenopus laevis oocytes by two electrode voltage-clamp electro...More data for this Ligand-Target Pair
TargetGlutamate receptor 3(Homo sapiens (Human))
Sibia Neurosciences

Curated by PDSP Ki Database
LigandPNGBDBM50060635((S)-2-Amino-3-(5-fluoro-2,4-dioxo-3,4-dihydro-2H-p...)
Affinity DataEC50:  2.09E+4nMAssay Description:Agonist activity at recombinant GluA3 receptor flip isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair