Affinity DataKi: 0.0450nMAssay Description:Displacement of [3H]AMPA from rat recombinant GluR3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 3(Homo sapiens (Human))
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 44.8nMAssay Description:Binding affinity for ionotropic Glutamate receptor AMPA 3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 3(Homo sapiens (Human))
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 1.80E+4nMAssay Description:Agonist activity at GluR3 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair