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Found 3 Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, NMDA 1' and Ligand = 'BDBM50078517'
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50078517(7-Nitro-4-oxo-4,5-dihydro-[1,2,4]triazolo[1,5-a]qu...)
Affinity DataKi:  710nMAssay Description:Binding affinity towards N-methyl-D-aspartate glutamate receptor 1 in rat cortical membranes using [3H]-glycine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50078517(7-Nitro-4-oxo-4,5-dihydro-[1,2,4]triazolo[1,5-a]qu...)
Affinity DataKi:  710nMAssay Description:Binding selectivity towards N-methyl-D-aspartate glutamate receptor 1 was determined by using [3H]- glycine/NMDAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50078517(7-Nitro-4-oxo-4,5-dihydro-[1,2,4]triazolo[1,5-a]qu...)
Affinity DataEC50:  7.80E+3nMAssay Description:Functional antagonism at the N-methyl-D-aspartate glutamate receptor 1 was demonstrated by the ability to inhibit the binding of thechannel-blocking ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed