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Found 2 Enz. Inhib. hit(s) with Target = 'Glutaminase kidney isoform, mitochondrial' and Ligand = 'BDBM50400063'
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University

US Patent
LigandPNGBDBM50400063(CHEMBL2177744 | US11191732, Example 4)
Affinity DataIC50:  4.60E+3nMAssay Description:A high throughput screening (HTS) assay and together with NCATS screened over 350,000 compounds in attempt to identify novel GLS inhibitor structures...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University

US Patent
LigandPNGBDBM50400063(CHEMBL2177744 | US11191732, Example 4)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of human kidney glutaminase (124 to 669) using L-[3H]-glutamine as substrate after 45 mins by GLS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed