Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Glutathione S-transferase P/Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) [T344D]' and Ligand = 'BDBM259282'
LigandPNGBDBM259282(US9499547, 23)
Affinity DataIC50:  18nMpH: 7.5 T: 2°CAssay Description:MKNK1-inhibitory activity at high ATP of compounds of the present invention after their preincubation with MKNK1 was quantified employing the TR-FRET...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent