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Found 2 Enz. Inhib. hit(s) with Target = 'Glycogen synthase kinase-3 beta' and Ligand = 'BDBM186202'
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandPNGBDBM186202(US9163013, 19)
Affinity DataIC50:  10nMT: 2°CAssay Description:Activity on human GSK-3beta was assessed using the following methods (according to Meijer et al., Chem. Biol., 2003-10:1255-1266).In a first screenin...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F.

US Patent
LigandPNGBDBM186202(US9163013, 19)
Affinity DataIC50:  12nMAssay Description:Inhibition of human recombinant GSK-3beta using Ulight-CFFKNIVTPRTPPPSQQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed