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Found 3 Enz. Inhib. hit(s) with Target = 'Glycogen synthase kinase-3 beta' and Ligand = 'BDBM50130724'
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50130724(1-(4-Amino-furazan-3-yl)-5-piperidin-1-ylmethyl-1H...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50130724(1-(4-Amino-furazan-3-yl)-5-piperidin-1-ylmethyl-1H...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Sterling Road

Curated by ChEMBL
LigandPNGBDBM50130724(1-(4-Amino-furazan-3-yl)-5-piperidin-1-ylmethyl-1H...)
Affinity DataEC50:  181nMAssay Description:Keywords: GSK3beta, dose response, kinase, inhibition, HTS Assay Overview: The glycogen synthase kinase-3 beta (GSK-3b) is a known master regulator f...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay