Found 3 Enz. Inhib. hit(s) with Target = 'Growth hormone secretagogue receptor type 1' and Ligand = 'BDBM19296'
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Univ Montpellier
Curated by ChEMBL
Univ Montpellier
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Displacement of red-ghrelin from SNAP-tagged human GHSR expressed in HEK293 cells incubated for 3 hrs at 4 degC or for 1 hr at room temperature by HT...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Univ Montpellier
Curated by ChEMBL
Univ Montpellier
Curated by ChEMBL
Affinity DataIC50: 32nM Kd: 19nMpH: 7.3 T: 2°CAssay Description:Specific binding was determined by incubation of membranes from GHS-R1a transfected LLC cells with 125I-His9-ghrelin in the presence of increasing co...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Univ Montpellier
Curated by ChEMBL
Univ Montpellier
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Displacement of 125I-[His9]-ghrelin from human GHSR1a expressed in LLC-PK1 cells by competitive binding assayMore data for this Ligand-Target Pair