Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with Target = 'Heat shock protein HSP 90-alpha' and Ligand = 'BDBM50533274'
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533274(Herbimycin C)
Affinity DataIC50:  17nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533274(Herbimycin C)
Affinity DataIC50:  17nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533274(Herbimycin C)
Affinity DataIC50:  18nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533274(Herbimycin C)
Affinity DataIC50:  18nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533274(Herbimycin C)
Affinity DataIC50:  18nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533274(Herbimycin C)
Affinity DataIC50:  18nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533274(Herbimycin C)
Affinity DataIC50:  20nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533274(Herbimycin C)
Affinity DataIC50:  20nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533274(Herbimycin C)
Affinity DataIC50:  22nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533274(Herbimycin C)
Affinity DataIC50:  22nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533274(Herbimycin C)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of HSP90alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed