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Found 10 Enz. Inhib. hit(s) with Target = 'Heat shock protein HSP 90-alpha' and Ligand = 'BDBM50533275'
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533275(CHEMBL4474732)
Affinity DataIC50:  53nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533275(CHEMBL4474732)
Affinity DataIC50:  53nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533275(CHEMBL4474732)
Affinity DataIC50:  56nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533275(CHEMBL4474732)
Affinity DataIC50:  56nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533275(CHEMBL4474732)
Affinity DataIC50:  57nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533275(CHEMBL4474732)
Affinity DataIC50:  57nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533275(CHEMBL4474732)
Affinity DataIC50:  59nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533275(CHEMBL4474732)
Affinity DataIC50:  59nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533275(CHEMBL4474732)
Affinity DataIC50:  65nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Peking Union Medical College & Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50533275(CHEMBL4474732)
Affinity DataIC50:  65nMAssay Description:Displacement of fluorescent labelled-VER00051001 from N-terminal ATP-binding site of human recombinant HSP90A expressed in Escherichia coli measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed