Found 8 Enz. Inhib. hit(s) with Target = 'Heat shock-related 70 kDa protein 2' and Ligand = 'BDBM50531165'
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research
Curated by ChEMBL
The Institute Of Cancer Research
Curated by ChEMBL
Affinity DataKi: <200nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 1 hr nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research
Curated by ChEMBL
The Institute Of Cancer Research
Curated by ChEMBL
Affinity DataKi: <200nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 1 hr nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research
Curated by ChEMBL
The Institute Of Cancer Research
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.33 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research
Curated by ChEMBL
The Institute Of Cancer Research
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.33 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research
Curated by ChEMBL
The Institute Of Cancer Research
Curated by ChEMBL
Affinity DataKi: 3.30E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.083 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research
Curated by ChEMBL
The Institute Of Cancer Research
Curated by ChEMBL
Affinity DataKi: 3.30E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) after 0.083 hrs nucleotide-derived FP probe displacement based by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research
Curated by ChEMBL
The Institute Of Cancer Research
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) assessed as initial inhibition constant nucleotide-derived FP probe displacement based by fluoresce...More data for this Ligand-Target Pair
TargetHeat shock-related 70 kDa protein 2(Homo sapiens)
The Institute Of Cancer Research
Curated by ChEMBL
The Institute Of Cancer Research
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Covalent inhibition of HSP72-NBD (unknown origin) assessed as initial inhibition constant nucleotide-derived FP probe displacement based by fluoresce...More data for this Ligand-Target Pair