Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Inverse agonist activity at human histamine H3 receptor by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair