Found 2 Enz. Inhib. hit(s) with Target = 'Inhibitor of nuclear factor kappa-B kinase subunit beta' and Ligand = 'BDBM50319741'
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 4.47E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair