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Found 4 Enz. Inhib. hit(s) with Target = 'Integrase' and Ligand = 'BDBM50486618'
TargetIntegrase(Human immunodeficiency virus 1)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50486618(CHEMBL2236600)
Affinity DataIC50:  250nMAssay Description:Inhibition of HIV-1 integrase assessed as inhibition of strand transfer activity using 32P-labeled DNA as substrate after 1 hr by gel-based assay in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50486618(CHEMBL2236600)
Affinity DataIC50: >1.23E+4nMAssay Description:Inhibition of HIV-1 integrase assessed as inhibition of 3'-processing activity using 32P-labeled DNA as substrate after 1 hr by gel-based assay in pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50486618(CHEMBL2236600)
Affinity DataIC50:  8.15E+7nMAssay Description:Inhibition of Human immunodeficiency virus 1 integrase 3'-processing activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetIntegrase(Human immunodeficiency virus 1)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50486618(CHEMBL2236600)
Affinity DataIC50:  2.50E+8nMAssay Description:Inhibition of Human immunodeficiency virus 1 integrase strand transfer activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article