Affinity DataKi: 130nMAssay Description:Displacement of [3H]diprenorphine from human kappa opioid receptor in CHO cells at 10 uMMore data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Displacement of [3H]diprenorphine from human kappa opioid receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Binding affinity against cloned human Opioid receptor kappa 1 using [125I]-D-Pro10-dynorphin A[1-11] as radioligandMore data for this Ligand-Target Pair