Affinity DataKi: 77nMAssay Description:Binding affinity against Opioid receptor kappa 1 using [3H]-U-69,593 as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 395nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 396nMAssay Description:Displacement of [3H]U-69593 from human recombinant Opioid receptor kappa 1 on CHO cell membranes.More data for this Ligand-Target Pair
Affinity DataKi: 515nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair