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Found 4 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50218796'
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Smithkline Beecham

Curated by ChEMBL
LigandPNGBDBM50218796(CHEMBL557978 | OXYMORPHINDOLE CHLORIDE | oxymorphi...)
Affinity DataKi:  77nMAssay Description:Binding affinity against Opioid receptor kappa 1 using [3H]-U-69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50218796(CHEMBL557978 | OXYMORPHINDOLE CHLORIDE | oxymorphi...)
Affinity DataKi:  395nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50218796(CHEMBL557978 | OXYMORPHINDOLE CHLORIDE | oxymorphi...)
Affinity DataKi:  396nMAssay Description:Displacement of [3H]U-69593 from human recombinant Opioid receptor kappa 1 on CHO cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50218796(CHEMBL557978 | OXYMORPHINDOLE CHLORIDE | oxymorphi...)
Affinity DataKi:  515nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed