TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California San Francisco
Curated by ChEMBL
University Of California San Francisco
Curated by ChEMBL
Affinity DataKi: 1.81E+3nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in membranes after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California San Francisco
Curated by ChEMBL
University Of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 1.70E+4nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293T assessed as intracellular cAMP accumulation after 15 mins by luciferase based GloSensor...More data for this Ligand-Target Pair