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Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50281761'
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50281761(CHEMBL4165704)
Affinity DataKi:  1.81E+3nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in membranes after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50281761(CHEMBL4165704)
Affinity DataEC50:  1.70E+4nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293T assessed as intracellular cAMP accumulation after 15 mins by luciferase based GloSensor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed