Found 2 Enz. Inhib. hit(s) with Target = 'Kynurenine--oxoglutarate transaminase 1' and Ligand = 'BDBM50324539'
TargetKynurenine--oxoglutarate transaminase 1(Homo sapiens (Human))
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant MBP-KAT1 expressed in HEK293 cells assessed as conversion of L-kynurenine to kynurenic acid after 1 hrMore data for this Ligand-Target Pair
TargetKynurenine--oxoglutarate transaminase 1(Homo sapiens (Human))
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of KAT1 in human prefrontal cortex homogenatesMore data for this Ligand-Target Pair