Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Legumain' and Ligand = 'BDBM22114'
TargetLegumain(Ixodes ricinus)
Georgia Institute of Technology

LigandPNGBDBM22114(aza-peptide Michael acceptor, 7a | ethyl (2E)-4-[(...)
Affinity DataIC50:  4.5nMT: 2°CAssay Description:AE activity in the induction medium was measured with the substrate Cbz-Ala-Ala-Asn-AMC. In a black 96-well microtiter plate, aza-peptidyl inhibitors...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Schistosoma mansoni)
Georgia Institute of Technology

LigandPNGBDBM22114(aza-peptide Michael acceptor, 7a | ethyl (2E)-4-[(...)
Affinity DataIC50:  31nMpH: 6.8 T: 2°CAssay Description:AE activity in the induction medium was measured with the substrate Cbz-Ala-Ala-Asn-AMC. In a black 96-well microtiter plate, aza-peptidyl inhibitors...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed