Found 4 Enz. Inhib. hit(s) with Target = 'Lysine-specific histone demethylase 1A' and Ligand = 'BDBM50582461'
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of recombinant LSD1 (157 to 852 residues) (unknown origin) expressed in Escherichia coli BL21 (DE) using H3K4me2 as substrate by amplex re...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of human LSD1 (unknown orgin)More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 1.64E+3nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Rabbit pulmonary artery(RPA) assay.More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Xinxiang Medical University
Curated by ChEMBL
Xinxiang Medical University
Curated by ChEMBL
Affinity DataKd: 240nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair