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Found 4 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50166529'
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50166529((+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazi...)
Affinity DataKi:  7.90nMAssay Description:Binding affinity for melanocortin-4 receptor transfected in HEK 293 cells using [125I]-NDP-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50166529((+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazi...)
Affinity DataIC50:  8.13nMAssay Description:Displacement of [125I]Nle4-D-Phe7-alpha-MSH from human MC4 receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50166529((+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazi...)
Affinity DataIC50:  8.13nMAssay Description:Displacement of [125I]Nle4-D-Phe7-alpha-MSH from human MC4 receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50166529((+/-)-1-[2-(4-fluorophenyl)-2-(4-isopropylpiperazi...)
Affinity DataIC50:  22nMAssay Description:Displacement of [125I]Nle4-D-Phe7-alpha-MSH from human MC4 receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed