Affinity DataIC50: 27nMAssay Description:Displacement of [125I][Nle4,D-Phe7]alpha-MSH from human MC5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Agonist activity at human MC5 receptor expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair