Found 3 Enz. Inhib. hit(s) with Target = 'Melanocyte-stimulating hormone receptor' and Ligand = 'BDBM50058158'
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 22.4nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataEC50: 2.61nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 1 receptorMore data for this Ligand-Target Pair