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Found 2 Enz. Inhib. hit(s) with Target = 'Melatonin receptor type 1B' and Ligand = 'BDBM50149169'
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50149169(CHEMBL127570 | Cyclopropanecarboxylic acid [3-(2-m...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity against human Melatonin receptor type 1B by using 2-[125I]-iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50149169(CHEMBL127570 | Cyclopropanecarboxylic acid [3-(2-m...)
Affinity DataEC50:  0.740nMAssay Description:Agonist activity of the compound was tested for its ability to inhibitforskolin-stimulated cAMP accumulation against MT receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed