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Found 4 Enz. Inhib. hit(s) with Target = 'Melatonin receptor type 1C' and Ligand = 'BDBM50470187'
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50470187(CHEMBL428882)
Affinity DataKi:  0.100nMAssay Description:Competitive binding by the displacement of 2-[125I]- Iodomelatonin binding from melatonin receptors in chicken brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50470187(CHEMBL428882)
Affinity DataKi:  0.100nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50470187(CHEMBL428882)
Affinity DataKi:  0.240nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50470187(CHEMBL428882)
Affinity DataEC50:  0.0370nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed