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Found 2 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 1' and Ligand = 'BDBM50252049'
TargetMetabotropic glutamate receptor 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252049((1S,3R)-1-aminopentane-1,3,5-tricarboxylic acid | ...)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat mGlu1 receptor expressed in HEK293 cells assessed as IP1 accumulation by IP-One functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252049((1S,3R)-1-aminopentane-1,3,5-tricarboxylic acid | ...)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat mGlu1 receptor expressed in HEK293 cells by intracellular Ca2+ mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed