Found 1 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 5' and Ligand = 'BDBM50429062'
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Brain Science Institute
Curated by ChEMBL
Brain Science Institute
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Antagonist activity at human mGluR5 expressed in HEK293 cells assessed as inhibition of L-glutamate-induced calcium mobilization by FDSS6000 assayMore data for this Ligand-Target Pair